Estrogen receptor modulator 1
CAS No. 63676-22-2
Estrogen receptor modulator 1 ( —— )
Catalog No. M24648 CAS No. 63676-22-2
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.46).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 61 | In Stock |
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10MG | 102 | In Stock |
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25MG | 169 | In Stock |
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50MG | 255 | In Stock |
|
100MG | 380 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameEstrogen receptor modulator 1
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NoteResearch use only, not for human use.
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Brief DescriptionEstrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.46).
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DescriptionEstrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.46).
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorEstrogen Receptor/ERR
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Research Area——
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Indication——
Chemical Information
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CAS Number63676-22-2
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Formula Weight242.3
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Molecular FormulaC14H10O2S
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESOC1=CC=C(C=C(C2=CC=C(O)C=C2)S3)C3=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Brogi S, et al. 3D-QSAR using pharmacophore-based alignment and virtual screening for discovery of novel MCF-7 cell line inhibitors. Eur J Med Chem. 2013 Sep;67:344-51.
molnova catalog
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